Organocatalytic Asymmetric Friedel–Crafts Reaction of Sesamol with Isatins: Access to Biologically Relevant 3-Aryl-3-hydroxy-2-oxindoles.

DOI Number:

10.1002/asia.201301546

Reaction Category:

RXNO ID:

RXNO_0000369

Educt:

sesamol, N-benzylisatin

Product:

(R)-1-Benzyl-3-hydroxy-3-(5-hydroxybenzo[d][1,3] dioxol-6-yl) indolin-2-one

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-(8α,9S)-cinchonan-9-ylthiourea

Cas No:

890044-38-9

Cas No:

485-71-2