Asymmetric vinylogous Mukaiyama aldol reaction of isatins under bifunctional organocatalysis: Enantioselective synthesis of substituted 3-hydroxy-2-oxindoles.

DOI Number:

10.1039/C8CC00759D

Reaction Category:

RXNO ID:

RXNO_0000016

Educt:

1-(4-(tert-butyl)benzyl)indoline-2,3-dione, (E)-(buta-1,3-dien-1-yloxy)trimethylsilane

Product:

substituted 3-hydroxy-2-oxindoles

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7

Associated Product from Buchler GmbH:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7