Organocatalytic tandem enantioselective Michael-cyclization of isatin-derived β,γ-unsaturated α-ketoesters with 3-hydroxy-4 h-chromen-4-one or 2-hydroxy-1, 4-naphthoquinone derivatives.

DOI Number:

10.1039/C6RA17400K

Reaction Category:

RXNO ID:

RXNO_0000009

Educt:

isatin-derived β,γ-unsaturated α-ketoesters, substituted 3-hydroxy-4H-chromen-4-one

Product:

spirocycles

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7

Associated Product from Buchler GmbH:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7