3-Alkyl-1,2,4-triazines as Heterocyclic Platforms for Organocatalytic Enantioselective Benzylic C–H Functionalization.

DOI Number:

10.1021/acs.orglett.5c00008

Reaction Category:

RXNO ID:

RXNO_0000009

Educt:

tert-butyl (Z)-2-cyano-2-(5-phenyl-1,2,4-triazin-3(2H)-ylidene)acetate, 4-hydroxy-4-methylpent-1-en-3-one

Product:

3-Alkyl-1,2,4-triazines

Catalyst:

3-[[3,5-bis(trifluoromethyl)phenyl]amino]-4-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1256245-84-7

Associated Product from Buchler GmbH:

3-[[3,5-bis(trifluoromethyl)phenyl]amino]-4-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1256245-84-7