Organocatalytic asymmetric Michael addition of benzofuran-2(3H)-ones to alkylideneindolenines generated in situ from arenesulfonylalkylindoles.

DOI Number:

10.1016/j.tetlet.2015.04.071

Reaction Category:

RXNO ID:

RXNO_0000009

Educt:

alkylideneindolenines, benzofuran-2(3H)-ones

Product:

substituted 3-((1H-indol-3-yl)methyl)benzofuran-2(3H)-one

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7

Associated Product from Buchler GmbH:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7