Bifunctional Thioureas Catalyzed Asymmetric Michael Addition of 1-Acetylindolin-3-ones to β,γ-Unsaturated α-Keto Esters.

DOI Number:

10.6023/cjoc201911027

Reaction Category:

RXNO ID:

RXNO_0000009

Educt:

1-acetylindolin-3-ones, β,γ-unsaturated α-keto esters

Product:

substituted ethyl (S)-2-oxo-4-(3-oxoindolin-2-yl)butanoate

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7

Associated Product from Buchler GmbH:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7