Catalytic asymmetric synthesis of α,β-disubstituted α,γ-diaminophosphonic acid precursors by michael addition of α-substituted nitrophosphonates to nitroolefins.

DOI Number:

10.1021/ol3012666

Reaction Category:

RXNO ID:

RXNO_0000009

Educt:

α-substituted nitrophosphonates, nitroolefins

Product:

diethyl ((2S,3R)-2-nitro-3-(nitromethyl)octan-2-yl)phosphonate

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7

Associated Product from Buchler GmbH:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7