Organocatalytic Activation of Diethyl Glutaconate for the Diastereo-and Enantioselective Assembly of NH-Free 2, 3, 4-Trisubstituted Pyrrolidines.

DOI Number:

10.1021/acs.orglett.7b00014

Reaction Category:

MOP ID:

MOP_0000561

Educt:

diethyl (E)-pent-2-enedioate, (E)-(2-nitrovinyl)benzene

Product:

ethyl (2R,3S,4R)-2-(2-ethoxy-2-oxoethyl)-4-phenylpyrrolidine-3-carboxylate

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7

Associated Product from Buchler GmbH:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7