Organocatalytic asymmetric intramolecular aza-Henry reaction: facile synthesis of trans-2,3-disubstituted tetrahydroquinolines.

DOI Number:

10.1039/C5OB00795J

Reaction Category:

RXNO ID:

RXNO_0000235

Educt:

substituted 2-(2-nitroethyl)aniline, aldehydes

Product:

trans-2,3-disubstituted tetrahydroquinolines

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7

Associated Product from Buchler GmbH:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7