Diversity-oriented enantioselective construction of atropisomeric heterobiaryls and N-aryl indoles via vinylidene ortho-quinone methides.

DOI Number:

10.31635/ccschem.021.202101154

Reaction Category:

Educt:

substituted (2-((2-hydroxynaphthalen-1-yl)ethynyl)phenyl)silanol, N-iodosuccinimide

Product:

atropisomeric heterobiaryls

Catalyst:

(2S)-2-[[[[3,5-bis(trifluoromethyl)phenyl]amino]thioxomethyl]amino]-N-[(8α,9S)-6′-methoxycinchonan-9-yl]-3-methyl-butanamide

Cas No:

1509940-71-9

Cas No:

130-95-0