Organocatalytic Enantioselective Construction of Chiral Azepine Skeleton Bearing Multiple‐Stereogenic Elements.

DOI Number:

10.1002/anie.202108040

Reaction Category:

MOP ID:

MOP_0000551

Educt:

1-((2-(9H-carbazol-9-yl)phenyl)ethynyl)naphthalen-2-ol, N-bromosuccinimide

Product:

azepine skeletons

Catalyst:

3-[[3,5-bis(trifluoromethyl)phenyl]amino]-4-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1256245-84-7

Associated Product from Buchler GmbH:

3-[[3,5-bis(trifluoromethyl)phenyl]amino]-4-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1256245-84-7