Asymmetric allylation by chiral organocatalyst‐promoted formal hetero‐Ene reactions of alkylgold intermediates.

DOI Number:

10.1002/anie.202012678

Reaction Category:

MOP ID:

MOP_0000561

Educt:

substituted N-(prop-2-yn-1-yl)formamide, substituted indoline-2,3-dione

Product:

substituted (R)-3-hydroxy-3-((S)-5-methylene-4,5-dihydrooxazol-4-yl)indolin-2-one

Catalyst:

3-[(3,5-dimethoxyphenyl)amino]-4-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

2579168-01-5

Cas No:

130-95-0