Highly Enantioselective Monofluoromethylation of C2-Arylindoles Using FBSM under Chiral Phase-Transfer Catalysis.

DOI Number:

10.1021/ol4013102

Reaction Category:

Educt:

phenyl(2-(p-tolyl)indolin-3-yl)methanesulfonyl tolyl, (fluoromethylenedisulfonyl)dibenzene

Product:

3-((S)-2-fluoro-1-phenyl-2,2-bis(phenylsulfonyl)ethyl)-2-(p-tolyl)indoline

Catalyst:

1-[[3,5-bis(1,1-dimethylethyl)phenyl]methyl]- 9-hydroxy-(9S)-Cinchonanium bromide (1:1)

Cas No:

1190864-60-8

Cas No:

118-10-5