Asymmetric sequential Au (I)/chiral tertiary amine catalysis: an enone-formation/cyanosilylation sequence to synthesize optically active 3-alkenyloxindoles from diazooxindoles.

DOI Number:

10.1039/C6CC00333H

Reaction Category:

MOP ID:

MOP_0000678

Educt:

diazooxindoles, 2,5-disubstituted furan, trimethylsilyl cyanide

Product:

3-alkenyloxindoles

Catalyst:

chloro(triphenylphosphine)gold, N-[3,5-bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-10,11-dihydro-6′-methoxy-cinchonan-9-yl]-Thiourea

Cas No:

852913-19-0

Cas No:

522-66-7