Catalyst-Controlled Switch in Diastereoselectivities: Enantioselective Construction of Functionalized 3,4-Dihydro-2H-thiopyrano[2,3-b]quinolines with Three Contiguous Stereocenters.

DOI Number:

10.1021/acs.joc.6b02688

Reaction Category:

Educt:

2-mercaptoquinoline-3-carbaldehydes, nitroolefins

Product:

3,4-Dihydro-2H-thiopyrano[2,3-b]quinolines

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7

Cas No:

852913-16-7