Cinchona alkaloid derivatives catalyzed asymmetric aza‐Friedel–crafts reaction of α‐naphthols with aryl aldimines.

DOI Number:

10.1002/chir.22714

Reaction Category:

RXNO ID:

RXNO_0000369

Educt:

1-Naphthol, 4-Methyl-N-[[2-(trifluoromethyl)phenyl]methylene]benzenesulfonamide

Product:

N-[(R)-(1-Hydroxy-2-naphthalenyl)[2-(trifluoromethyl)phenyl]methyl]-4-methylbenzenesulfonamide

Catalyst:

4-((R)-((tert-butyldiphenylsilyl)oxy)((1S,2S,4S,5R)- 5-vinylquinuclidin-2-yl)methyl)quinolin-6-ol

Cas No:

Cas No:

524-63-0