Direct catalytic asymmetric synthesis of oxindole-derived δ-hydroxy-β-ketoesters by Aldol reactions.

DOI Number:

10.1021/acs.orglett.9b03527

Reaction Category:

RXNO ID:

RXNO_0000016

Educt:

5-methoxyindoline-2,3-dione, methyl 3-oxobutanoate

Product:

methyl (R)-4-(3-hydroxy-5-methoxy-2-oxoindolin-3-yl)-3-oxobutanoate

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(9R)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-25-8

Associated Product from Buchler GmbH:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(9R)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-25-8