Bifuctional amino-squaramides catalyzed asymmetric spiroannulation cascades with aliphatic β, γ-unsaturated α-keto esters: controlling an aldehyde enolate.

DOI Number:

10.1021/jo202633c

Reaction Category:

RXNO ID:

RXNO_0000009

Educt:

2-oxocyclohexane-1-carbaldehyde, aliphatic beta,gamma-unsaturated α-keto esters

Product:

substituted (6R)-1,7-dioxo-2-oxaspiro[5.5]undecane-3-carboxylate

Catalyst:

3-[[[3,5-bis(trifluoromethyl)phenyl]methyl]amino]-4-[[(9R)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1362169-08-1

Cas No:

56-54-2