Highly Enantioselective Dihydroxylation of 1,1-Disubstituted Aliphatic Alkenes Enabled by Orchestrated Noncovalent π-Interactions.

DOI Number:

10.1021/acs.orglett.3c04188

Reaction Category:

MOP ID:

MOP_0000673

Educt:

1,1-disubstituted aliphatic alkenes

Product:

(R)-2-methyl-3-((4-(3,4,5-trimethoxyphenyl)phthalazin-1-yl)oxy)propane-1,2-diol

Catalyst:

dipotassium osmate, (8α,9R)-(8′′α,9′′R)-9,9′′-[1,4-Phthalazinediylbis (oxy)]bis[10,11-dihydro-6′-methoxycinchonan]

Cas No:

140924-50-1

Associated Product from Buchler GmbH:

1,4-Bis(9-O-dihydroquininyl)phthalazine (DHQ)2PHAL

Cas No:

140924-50-1