Stereoselective organocatalytic sulfa-Michael reactions of aryl substituted α,β-unsaturated N-acyl pyrazoles.

DOI Number:

10.1039/C8QO00357B

Reaction Category:

RXNO ID:

RXNO_0000009

Educt:

aryl substituted α,β-unsaturated N-acyl pyrazoles, benzenethiol

Product:

(R)-3-cyclohexyl-3-(phenylthio)-1-(1H-pyrazol-1-yl)propan-1-one

Catalyst:

3-[[3,5-Bis(trifluoromethyl)phenyl]amino]-4-[[(8α,9S)-10,11-dihydro-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1352957-59-5

Cas No:

522-66-7