Organocatalytic Enantioselective Aminoalkylation of 5‐Aminopyrazole Derivatives with Cyclic Imines.

DOI Number:

10.1002/ejoc.202001314

Reaction Category:

MOP ID:

MOP_0000369

Educt:

cyclic imines, 5‐aminopyrazoles

Product:

substituted (S)-4-(5-amino-1H-pyrazol-4-yl)-3,4-dihydrobenzo[e][1,2,3]oxathiazine 2,2-dioxide

Catalyst:

3-[(1,1-dimethylethyl)amino]-4-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1610724-48-5

Cas No:

130-95-0