Supramolecular catalysis in the dearomative Michael addition involving nitro-group-activated benzofurans.

DOI Number:

10.1039/D5QO00035A

Reaction Category:

RXNO ID:

RXNO_0000009

Educt:

nitro-group-activated benzofurans, 5-phenylfuranone

Product:

(R)-5-((2R,3S)-2-nitro-2,3-dihydrobenzofuran-3-yl)-5-phenylfuran-2(5H)-one

Catalyst:

3-[[3,5-bis(trifluoromethyl)phenyl]amino]-4-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1256245-84-7

Associated Product from Buchler GmbH:

3-[[3,5-bis(trifluoromethyl)phenyl]amino]-4-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1256245-84-7