Chiral synthetic unprecedented spiro [indoline-2,3′-thiophen]-3-ones via an organocatalytic asymmetric sulfa-Michael/aldol cascade reaction.

DOI Number:

10.1039/D4QO01551G

Reaction Category:

Educt:

substituted indolin-3-one, 2,5-disubstituted 1,4-dithiane-2,5-diol

Product:

spiro [indoline-2,3′-thiophen]-3-ones

Catalyst:

3-[[3,5-bis(trifluoromethyl)phenyl]amino]-4-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1256245-84-7

Associated Product from Buchler GmbH:

3-[[3,5-bis(trifluoromethyl)phenyl]amino]-4-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1256245-84-7